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Apixaban MR2 — Competitive Intelligence Brief
phase 1
Factor Xa inhibitor
Factor Xa
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Apixaban MR2 (Apixaban MR2) — Pfizer. Factor Xa inhibitor
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Apixaban MR2 TARGET | Apixaban MR2 | Pfizer | phase 1 | Factor Xa inhibitor | Factor Xa | |
| Hympavzi | MARSTACIMAB | Pfizer Inc | marketed | Monoclonal Antibody | Factor Xa | 2025-01-01 |
| Eliquis | apixaban | Bristol-Myers Squibb | marketed | Factor Xa inhibitor | Factor Xa (FXa) | 2012-01-01 |
| Xarelto | rivaroxaban | Johnson & Johnson | marketed | Direct Factor Xa Inhibitor | Factor Xa (FXa) | 2011-01-01 |
| Heparin Sodium In Plastic Container | Heparin Sodium | Fresenius Kabi | marketed | Anti-coagulant | Antithrombin III, Factor Xa, Factor IIa | 1939-01-01 |
| Fondaparinux Sodium (Arixtra) | Fondaparinux Sodium (Arixtra) | Paul Di Cesare,MD | marketed | Factor Xa inhibitor | Factor Xa | |
| Apixaban 2.5 milligram | Apixaban 2.5 milligram | McMaster University | marketed | Direct Factor Xa inhibitor | Factor Xa |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Factor Xa inhibitor class)
- GlaxoSmithKline · 4 drugs in this class
- Bayer · 2 drugs in this class
- China National Center for Cardiovascular Diseases · 1 drug in this class
- Hoffmann-La Roche · 1 drug in this class
- Kim, Seok Jin · 1 drug in this class
- NYU Langone Health · 1 drug in this class
- Paul Di Cesare,MD · 1 drug in this class
- Pfizer · 1 drug in this class
- Queen Mary University of London · 1 drug in this class
- Queen's University · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Apixaban MR2 — Competitive Intelligence Brief. https://druglandscape.com/ci/apixaban-mr2. Accessed 2026-05-13.
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