Last reviewed · How we verify
APD356 — Competitive Intelligence Brief
phase 2
CB2 receptor agonist
CB2
Neurology
Small molecule
Live · refreshed every 30 min
Target snapshot
APD356 (APD356) — Eisai Inc.. APD356 is a selective agonist of the cannabinoid receptor type 2 (CB2).
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| APD356 TARGET | APD356 | Eisai Inc. | phase 2 | CB2 receptor agonist | CB2 | |
| CBD | CBD | Stero Biotechs Ltd. | marketed | Cannabinoid | 5-HT1A, TRPV1, GPR55, CB1 (allosteric), CB2 (allosteric) | |
| MediCabilis CBD Oil | MediCabilis CBD Oil | Gold Coast Hospital and Health Service | marketed | Cannabinoid | CB1 receptor, CB2 receptor, 5-HT1A receptor, TRPV1 receptor (multiple targets) | |
| Cannabis Extract Oil SR Capsule | Cannabis Extract Oil SR Capsule | University of Sao Paulo General Hospital | marketed | Cannabinoid receptor modulator | CB1 receptor, CB2 receptor | |
| Cannabis Sativa Oil | Cannabis Sativa Oil | Fondation pour l'accueil et l'hébérement des personnes âgées | marketed | Phytocannabinoid preparation | CB1 receptor, CB2 receptor | |
| Cesamet™ (nabilone) | Cesamet™ (nabilone) | NEMA Research, Inc. | marketed | Synthetic cannabinoid | CB1 and CB2 cannabinoid receptors | |
| Cannabis oil | Cannabis oil | Assaf-Harofeh Medical Center | marketed | Phytocannabinoid preparation | CB1 receptor, CB2 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (CB2 receptor agonist class)
- Creabilis SA · 1 drug in this class
- Eisai Inc. · 1 drug in this class
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Cite this brief
Drug Landscape (2026). APD356 — Competitive Intelligence Brief. https://druglandscape.com/ci/apd356. Accessed 2026-05-14.
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