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Apalutamide Oral Tablet — Competitive Intelligence Brief

Apalutamide Oral Tablet (Apalutamide Oral Tablet) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Androgen receptor antagonist. Area: Oncology.

phase 3 Androgen receptor antagonist Androgen receptor (AR) Oncology Small molecule Live · refreshed every 30 min

Target snapshot

Apalutamide Oral Tablet (Apalutamide Oral Tablet) — Santa Chiara Hospital. Apalutamide is an androgen receptor inhibitor that blocks the binding and nuclear translocation of androgens, preventing androgen-driven prostate cancer cell growth.

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
Apalutamide Oral Tablet TARGET Apalutamide Oral Tablet Santa Chiara Hospital phase 3 Androgen receptor antagonist Androgen receptor (AR)
ODM-201 Tablet A ODM-201 Tablet A Orion Corporation, Orion Pharma marketed Androgen receptor antagonist Androgen receptor (AR)
Zoladex and Casodex Zoladex and Casodex AstraZeneca marketed GnRH agonist (Zoladex) and androgen receptor antagonist (Casodex) GnRH receptor (Zoladex); androgen receptor (Casodex)
Darolutamide Oral Tablet Darolutamide Oral Tablet Santa Chiara Hospital marketed Androgen receptor antagonist Androgen receptor (AR)
Maximum androgen blockade Maximum androgen blockade Wonju Severance Christian Hospital marketed Androgen receptor antagonist combination therapy Androgen receptor; testosterone synthesis pathway
Darolutamide continuous Darolutamide continuous The First Affiliated Hospital with Nanjing Medical University phase 3 Androgen receptor antagonist Androgen receptor (AR)
Enzalutamide Soft Capsules Enzalutamide Soft Capsules Jiangsu HengRui Medicine Co., Ltd. phase 3 Androgen receptor antagonist Androgen receptor (AR)

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Androgen receptor antagonist class)

  1. Santa Chiara Hospital · 2 drugs in this class
  2. Cassiopea SpA · 2 drugs in this class
  3. The First Affiliated Hospital with Nanjing Medical University · 2 drugs in this class
  4. Pfizer · 2 drugs in this class
  5. Suzhou Kintor Pharmaceutical Inc, · 1 drug in this class
  6. AEterna Zentaris · 1 drug in this class
  7. University of Sydney · 1 drug in this class
  8. CHU de Quebec-Universite Laval · 1 drug in this class
  9. Jiangsu HengRui Medicine Co., Ltd. · 1 drug in this class
  10. Orion Corporation, Orion Pharma · 1 drug in this class

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Cite this brief

Drug Landscape (2026). Apalutamide Oral Tablet — Competitive Intelligence Brief. https://druglandscape.com/ci/apalutamide-oral-tablet. Accessed 2026-05-14.

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