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Aliskiren 150 — Competitive Intelligence Brief
phase 3
Direct renin inhibitor
Renin
Cardiovascular
Small molecule
Live · refreshed every 30 min
Target snapshot
Aliskiren 150 (Aliskiren 150) — Novartis. Aliskiren is a direct renin inhibitor that blocks the first step of the renin-angiotensin-aldosterone system (RAAS) by preventing renin from converting angiotensinogen to angiotensin I.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| Aliskiren 150 TARGET | Aliskiren 150 | Novartis | phase 3 | Direct renin inhibitor | Renin | |
| Tekturna | ALISKIREN | Lxo Ireland | marketed | Renin Inhibitor | Renin | 2007-01-01 |
| Capozide 25/15 | CAPTOPRIL | Aarxion Anda Hlding | marketed | Thiazide Diuretic [EPC] | Renin | 1981-01-01 |
| Keverprazan 14 days | Keverprazan 14 days | Second Affiliated Hospital, School of Medicine, Zhejiang University | marketed | direct renin inhibitor | renin | |
| Aliskiren, Perindopril | Aliskiren, Perindopril | Medical University of Gdansk | marketed | Antihypertensive combination (direct renin inhibitor + ACE inhibitor) | Renin and Angiotensin-Converting Enzyme (ACE) | |
| Valsartan/aliskiren | Valsartan/aliskiren | Novartis | marketed | Angiotensin II receptor blocker + direct renin inhibitor combination | AT1 receptor (valsartan); renin (aliskiren) | |
| Aliskiren + Valsartan | Aliskiren + Valsartan | HeartDrug Research LLC | marketed | Direct renin inhibitor + angiotensin II receptor blocker combination | Renin and AT1 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Direct renin inhibitor class)
- Medical Practice Prof D. Ivanov · 1 drug in this class
- Novartis · 1 drug in this class
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Cite this brief
Drug Landscape (2026). Aliskiren 150 — Competitive Intelligence Brief. https://druglandscape.com/ci/aliskiren-150. Accessed 2026-06-10.
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