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14C-paliperidone — Competitive Intelligence Brief

14C-paliperidone (14C-paliperidone) competitive landscape: 6 comparators, recent regulatory actions, upcoming PDUFA, patent timeline. Class: Atypical antipsychotic. Area: Neurology.

phase 1 Atypical antipsychotic Dopamine D2 receptor Neurology Small molecule Live · refreshed every 30 min

Target snapshot

14C-paliperidone (14C-paliperidone) — Johnson & Johnson Pharmaceutical Research & Development, L.L.C.. Dopamine D2 receptor antagonist

Comparator set (6 drugs)

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DrugGenericSponsorPhaseClassTargetApproval / PDUFA
14C-paliperidone TARGET 14C-paliperidone Johnson & Johnson Pharmaceutical Research & Development, L.L.C. phase 1 Atypical antipsychotic Dopamine D2 receptor
Aripiprazole tablet Aripiprazole tablet All India Institute of Medical Sciences, Bhubaneswar marketed Atypical antipsychotic Dopamine D2 receptor (partial agonist); Serotonin 5-HT1A receptor (partial agonist); Serotonin 5-HT2A receptor (antagonist)
Risperidone and Ramelteon Risperidone and Ramelteon All India Institute of Medical Sciences, Bhubaneswar marketed Atypical antipsychotic + melatonin receptor agonist combination Dopamine D2 receptor, serotonin 5-HT2A receptor, melatonin MT1/MT2 receptors
Quetiapine (drug) Quetiapine (drug) Medical University of Vienna marketed Atypical antipsychotic Dopamine D2 receptor, Serotonin 5-HT2A receptor
Aripiprazole; Quetiapine Aripiprazole; Quetiapine Taichung Veterans General Hospital marketed Atypical antipsychotic combination Dopamine D2 receptor; Serotonin 5-HT2A receptor; Serotonin 5-HT1A receptor
Lithium carbonate + perospirone hydrochloride Lithium carbonate + perospirone hydrochloride Shanghai Mental Health Center marketed Mood stabilizer + atypical antipsychotic combination Inositol monophosphatase, GSK-3 (lithium); dopamine D2 receptor, serotonin 5-HT2A receptor (perospirone)
sodium valproate with Clozapine sodium valproate with Clozapine Shanghai Mental Health Center marketed Antipsychotic + mood stabilizer combination Dopamine D2 receptor, serotonin 5-HT2A receptor, GABA pathways, histone deacetylase

Recent regulatory actions (last 90 days)

No regulatory actions in the last 90 days for this set.

Upcoming PDUFA dates (next 180 days)

No PDUFA dates in the next 180 days for this set.

Patent timeline (forward window)

No upcoming patent expiries for this set.

Sponsor landscape (Atypical antipsychotic class)

  1. Shanghai Mental Health Center · 10 drugs in this class
  2. AstraZeneca · 6 drugs in this class
  3. Otsuka Pharmaceutical Development & Commercialization, Inc. · 5 drugs in this class
  4. Johnson & Johnson Pharmaceutical Research & Development, L.L.C. · 4 drugs in this class
  5. Eli Lilly and Company · 4 drugs in this class
  6. Otsuka Pharmaceutical Co., Ltd. · 3 drugs in this class
  7. Medical University of Vienna · 2 drugs in this class
  8. Organon and Co · 2 drugs in this class
  9. Chengdu Kanghong Pharmaceutical Group Co., Ltd. · 2 drugs in this class
  10. H. Lundbeck A/S · 2 drugs in this class

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Cite this brief

Drug Landscape (2026). 14C-paliperidone — Competitive Intelligence Brief. https://druglandscape.com/ci/14c-paliperidone. Accessed 2026-06-10.

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Primary sources · FDA · ClinicalTrials.gov · EMA · SEC EDGAR · ChEMBL · Wikidata · full sourcing