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[11C]raclopride — Competitive Intelligence Brief
marketed
Dopamine D2/D3 receptor antagonist (PET imaging agent)
Dopamine D2 receptor, Dopamine D3 receptor
Neurology, Psychiatry, Medical Imaging
Small molecule
Live · refreshed every 30 min
Target snapshot
[11C]raclopride ([11C]raclopride) — New York State Psychiatric Institute. [11C]raclopride is a radioactive dopamine D2/D3 receptor antagonist used as a positron emission tomography (PET) imaging agent to visualize dopamine receptor binding in the brain.
Comparator set (6 drugs)
| Drug | Generic | Sponsor | Phase | Class | Target | Approval / PDUFA |
|---|---|---|---|---|---|---|
| [11C]raclopride TARGET | [11C]raclopride | New York State Psychiatric Institute | marketed | Dopamine D2/D3 receptor antagonist (PET imaging agent) | Dopamine D2 receptor, Dopamine D3 receptor | |
| Ropinirole (Requip) | Ropinirole (Requip) | St. Luke's-Roosevelt Hospital Center | marketed | Dopamine D2/D3 receptor agonist | Dopamine D2 receptor, Dopamine D3 receptor | |
| Amisulpride add-on | Amisulpride add-on | National Health Research Institutes, Taiwan | marketed | Atypical antipsychotic | Dopamine D2 receptor, Dopamine D3 receptor | |
| Raclopride C11 | Raclopride C11 | University of North Carolina, Chapel Hill | marketed | Dopamine D2/D3 receptor antagonist (PET imaging agent) | Dopamine D2 receptor, Dopamine D3 receptor | |
| IM aripiprazole once monthly | IM aripiprazole once monthly | University of Utah | marketed | Atypical antipsychotic | Dopamine D2 receptor, Dopamine D3 receptor | |
| aripiprazole long acting injectable formulation | aripiprazole long acting injectable formulation | Vanguard Research Group | marketed | Atypical antipsychotic (dopamine partial agonist) | Dopamine D2 receptor, Dopamine D3 receptor | |
| ropinirole CR-RLS | ropinirole CR-RLS | GlaxoSmithKline | marketed | Dopamine D2/D3 receptor agonist | Dopamine D2 receptor, Dopamine D3 receptor |
Recent regulatory actions (last 90 days)
Upcoming PDUFA dates (next 180 days)
Patent timeline (forward window)
Sponsor landscape (Dopamine D2/D3 receptor antagonist (PET imaging agent) class)
- New York State Psychiatric Institute · 1 drug in this class
- University of North Carolina, Chapel Hill · 1 drug in this class
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Cite this brief
Drug Landscape (2026). [11C]raclopride — Competitive Intelligence Brief. https://druglandscape.com/ci/11c-raclopride. Accessed 2026-05-16.
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