{"id":"inaperisone","rwe":[{"pmid":"16126840","year":"2005","title":"Tolperisone-type drugs inhibit spinal reflexes via blockade of voltage-gated sodium and calcium channels.","finding":"","journal":"The Journal of pharmacology and experimental therapeutics","studyType":"Clinical Study"},{"pmid":"10812055","year":"2000","title":"Effects of TAK-637, a tachykinin receptor antagonist, on the micturition reflex in guinea pigs.","finding":"","journal":"European journal of pharmacology","studyType":"Clinical Study"},{"pmid":"10594323","year":"1999","title":"Effects of TAK-637, a tachykinin receptor antagonist, on lower urinary tract function in the guinea pig.","finding":"","journal":"European journal of pharmacology","studyType":"Clinical Study"},{"pmid":"1618281","year":"1992","title":"Inhibitory effect of inaperisone hydrochloride (inaperisone), a new centrally acting muscle relaxant, on the micturition reflex.","finding":"","journal":"European journal of pharmacology","studyType":"Clinical Study"},{"pmid":"1785387","year":"1991","title":"[Identification of effective region of the pons in response to inaperisone which facilitates urine storage].","finding":"","journal":"Hinyokika kiyo. Acta urologica Japonica","studyType":"Clinical Study"}],"tags":[{"label":"Small Molecule","category":"modality"},{"label":"Active","category":"status"}],"phase":"phase_2","safety":{},"trials":[],"aliases":[],"patents":[],"pricing":[],"allNames":"(+/-)-inaperisone","offLabel":[],"synonyms":["inaperisone hydrochloride","inaperisone HCl","inaperisone","(+/-)-Inaperisone"],"timeline":[],"approvals":[],"brandName":"(+/-)-Inaperisone","ecosystem":[],"mechanism":{"modality":"Small Molecule","explanation":"Imagine INAPERISONE as a key that fits into a lock in the body. When it binds to this lock, it triggers a series of events that help to treat a particular condition. This process is complex and involves many different molecules and pathways, but essentially, INAPERISONE helps to restore balance and normal function to the body.","oneSentence":"INAPERISONE is thought to work by interacting with a specific target in the body to produce a therapeutic effect.","technicalDetail":"INAPERISONE is a small molecule that modulates the activity of a specific protein or receptor, leading to a cascade of downstream effects that ultimately result in its therapeutic effects."},"commercial":{},"references":[{"id":1,"url":"https://drugcentral.org/drugcard/3297","fields":["approvals","synonyms","ATC","PK","indications","contraindications","DDIs","targets","patents","FAERS"],"source":"DrugCentral"},{"id":2,"url":"https://pubmed.ncbi.nlm.nih.gov/?term=INAPERISONE","fields":["publications"],"source":"PubMed/NCBI"}],"_enrichedAt":"2026-03-30T12:03:30.427835","biosimilars":[],"competitors":[],"genericName":"inaperisone","indications":{"approved":[],"offLabel":[],"pipeline":[]},"drugCategory":"active","labelChanges":[],"relatedDrugs":[],"trialDetails":[],"genericFilers":[],"latestUpdates":[],"manufacturing":[],"crossReferences":{"UNII":"0QAC3P785O","CHEBI":"CHEBI:134999","INN_ID":"6262","UMLSCUI":"C0062996","ChEMBL_ID":"CHEMBL1797127","PUBCHEM_CID":"65860","SECONDARY_CAS_RN":"118230-97-0","MESH_SUPPLEMENTAL_RECORD_UI":"C052425"},"formularyStatus":[],"_enricherVersion":"v2","developmentCodes":[],"ownershipHistory":[],"publicationCount":6,"therapeuticAreas":["Other"],"biosimilarFilings":[],"recentPublications":[{"date":"2005 Dec","pmid":"16126840","title":"Tolperisone-type drugs inhibit spinal reflexes via blockade of voltage-gated sodium and calcium channels.","journal":"The Journal of pharmacology and experimental therapeutics"},{"date":"2000 May 3","pmid":"10812055","title":"Effects of TAK-637, a tachykinin receptor antagonist, on the micturition reflex in guinea pigs.","journal":"European journal of pharmacology"},{"date":"1999 Nov 3","pmid":"10594323","title":"Effects of TAK-637, a tachykinin receptor antagonist, on lower urinary tract function in the guinea pig.","journal":"European journal of pharmacology"},{"date":"1992 Mar 31","pmid":"1618281","title":"Inhibitory effect of inaperisone hydrochloride (inaperisone), a new centrally acting muscle relaxant, on the micturition reflex.","journal":"European journal of pharmacology"},{"date":"1991 Dec","pmid":"1785387","title":"[Identification of effective region of the pons in response to inaperisone which facilitates urine storage].","journal":"Hinyokika kiyo. Acta urologica Japonica"}],"companionDiagnostics":[],"genericManufacturerList":[],"status":"active","companyName":"","companyId":"","modality":"Small molecule","firstApprovalDate":"","aiSummary":"(+/-)-Inaperisone is a small molecule. It is also known by the synonyms INAPERISONA and INAPERISONE.","enrichmentLevel":3,"visitCount":0,"trialStats":{"total":0,"withResults":0},"verificationStatus":"partial","dataCompleteness":{"mechanism":true,"indications":false,"safety":false,"trials":false,"score":1}}