{"id":"f-choline-intravenous-injection","safety":{"commonSideEffects":[{"rate":null,"effect":"Radiation exposure"},{"rate":null,"effect":"Injection site reactions"}]},"_chembl":null,"_dailymed":null,"mechanism":{"_ai_source":"claude-haiku-4.5","explanation":"F-choline accumulates in cells with high choline uptake and metabolism, particularly in tumors and areas of inflammation. The fluorine-18 radiolabel allows detection via PET imaging, enabling visualization of metabolically active lesions. This is used primarily for oncologic imaging to detect and stage malignancies.","oneSentence":"F-choline is a fluorine-18 labeled choline analog used as a positron emission tomography (PET) imaging agent to visualize choline metabolism in tissues.","_ai_confidence":"medium"},"_scrapedAt":"2026-03-28T01:12:09.370Z","_scrapedBy":"cloudflare-swarm","_wikipedia":null,"indications":{"approved":[{"name":"PET imaging of prostate cancer"},{"name":"PET imaging of other malignancies with elevated choline metabolism"}]},"trialDetails":[{"nctId":"NCT04999215","phase":"PHASE3","title":"Choline-PET: Exploratory Study Assessing the Potential Role of F-choline PET Imaging in New and Emerging Indications","status":"RECRUITING","sponsor":"Centre hospitalier de l'Université de Montréal (CHUM)","startDate":"2022-08-01","conditions":"Lesion With Known or Suspected F-choline Uptake","enrollment":500}],"_emaApprovals":[],"_faersSignals":[],"_approvalHistory":[],"publicationCount":4,"rwe":[],"genericFilers":[],"relatedDrugs":[],"labelChanges":[],"biosimilarFilings":[],"pricing":[],"formularyStatus":[],"manufacturing":[],"companionDiagnostics":[],"competitors":[],"timeline":[],"patents":[],"ownershipHistory":[],"trials":[],"biosimilars":[],"latestUpdates":[],"references":[],"tags":[],"ecosystem":[],"genericManufacturerList":[],"offLabel":[],"developmentCodes":[],"aliases":["Fluorocholine"],"phase":"phase_3","status":"active","brandName":"F-choline intravenous injection","genericName":"F-choline intravenous injection","companyName":"Centre hospitalier de l'Université de Montréal (CHUM)","companyId":"centre-hospitalier-de-l-universit-de-montr-al-chum","modality":"Small molecule","firstApprovalDate":"","aiSummary":"F-choline is a fluorine-18 labeled choline analog used as a positron emission tomography (PET) imaging agent to visualize choline metabolism in tissues. Used for PET imaging of prostate cancer, PET imaging of other malignancies with elevated choline metabolism.","enrichmentLevel":3,"visitCount":1,"trialStats":{"total":1,"withResults":0},"verificationStatus":"verified","dataCompleteness":{"mechanism":true,"indications":true,"safety":true,"trials":true,"score":4}}