{"id":"domitroban","rwe":[],"tags":[{"label":"domitroban","category":"class"},{"label":"Small Molecule","category":"modality"},{"label":"Thromboxane A2 receptor","category":"target"},{"label":"TBXA2R","category":"gene"},{"label":"Active","category":"status"}],"phase":"phase_2","safety":{},"trials":[],"aliases":[],"patents":[],"pricing":[],"allNames":["domitroban","domitroban calcium","domitroban calcium hydrate"],"offLabel":[],"synonyms":["domitroban","domitroban calcium","domitroban calcium hydrate"],"timeline":[],"aiSummary":"DOMITROBAN is a small molecule drug that targets the thromboxane A2 receptor. It is classified as a domitroban, but its commercial status and approved indications are unknown. DOMITROBAN works by inhibiting the action of thromboxane A2, a substance that promotes blood clotting. As a result, it may be used to treat conditions related to excessive blood clotting, although its specific indications are not specified. Further information on its development, approval, and safety profile is needed.","approvals":[],"ecosystem":[],"mechanism":{"target":"Thromboxane A2 receptor, Thromboxane A2 receptor","targets":[{"gene":"TBXA2R","source":"DrugCentral","target":"Thromboxane A2 receptor","protein":"Thromboxane A2 receptor"}],"modality":"Small Molecule","drugClass":"domitroban","explanation":"Think of thromboxane A2 like a messenger that tells blood cells to stick together and form clots. DOMITROBAN acts like a 'blocker' that prevents this messenger from doing its job, which can help prevent unwanted blood clots from forming.","oneSentence":"DOMITROBAN blocks the action of thromboxane A2, a substance that promotes blood clotting.","technicalDetail":"DOMITROBAN is a thromboxane A2 receptor antagonist, which means it binds to and blocks the action of the thromboxane A2 receptor, a G-protein coupled receptor involved in platelet activation and aggregation."},"commercial":{},"references":[{"id":1,"url":"https://drugcentral.org/drugcard/3165","fields":["approvals","synonyms","ATC","PK","indications","contraindications","DDIs","targets","patents","FAERS"],"source":"DrugCentral"},{"id":2,"url":"https://pubmed.ncbi.nlm.nih.gov/?term=DOMITROBAN","fields":["publications"],"source":"PubMed/NCBI"}],"_enrichedAt":"2026-03-30T10:49:09.448714","biosimilars":[],"competitors":[{"drugName":"dinoprost","drugSlug":"dinoprost","fdaApproval":"1976-05-18","patentStatus":"Unknown","relationship":"same-target"},{"drugName":"dinoprostone","drugSlug":"dinoprostone","fdaApproval":"1977-08-23","patentStatus":"Unknown","relationship":"same-target"},{"drugName":"iloprost","drugSlug":"iloprost","fdaApproval":"2004-12-29","patentExpiry":"Jul 18, 2044","patentStatus":"Patent protected","relationship":"same-target"},{"drugName":"losartan","drugSlug":"losartan","fdaApproval":"1995-04-14","patentExpiry":"Oct 7, 2041","patentStatus":"Patent protected","relationship":"same-target"}],"dataSources":[{"url":"https://drugcentral.org","name":"DrugCentral","fields":["indications","contraindications","safety","target","drugInteractions"],"retrievedDate":"2026-04-07"}],"genericName":"domitroban","indications":{"approved":[],"offLabel":[],"pipeline":[]},"drugCategory":"active","labelChanges":[],"relatedDrugs":[{"drugId":"dinoprost","brandName":"dinoprost","genericName":"dinoprost","approvalYear":"1976","relationship":"same-target"},{"drugId":"dinoprostone","brandName":"dinoprostone","genericName":"dinoprostone","approvalYear":"1977","relationship":"same-target"},{"drugId":"iloprost","brandName":"iloprost","genericName":"iloprost","approvalYear":"2004","relationship":"same-target"},{"drugId":"losartan","brandName":"losartan","genericName":"losartan","approvalYear":"1995","relationship":"same-target"}],"trialDetails":[],"genericFilers":[],"latestUpdates":[],"manufacturing":[],"administration":{},"crossReferences":{"UNII":"742F5K270Q","CHEBI":"CHEBI:135586","INN_ID":"7348","UMLSCUI":"C1880393","ChEMBL_ID":"CHEMBL3301671","KEGG_DRUG":"D09824","PUBCHEM_CID":"5312138","IUPHAR_LIGAND_ID":"1979"},"formularyStatus":[],"_enricherVersion":"v2","developmentCodes":[],"ownershipHistory":[],"publicationCount":0,"therapeuticAreas":["Cardiovascular"],"biosimilarFilings":[],"recentPublications":[],"companionDiagnostics":[],"genericManufacturerList":[],"status":"active","brandName":"DOMITROBAN","companyName":"","companyId":"","modality":"Small molecule","firstApprovalDate":"","enrichmentLevel":3,"visitCount":0,"trialStats":{"total":0,"withResults":0},"verificationStatus":"partial","dataCompleteness":{"mechanism":true,"indications":false,"safety":false,"trials":false,"score":1}}